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Pentobarbital, also known as pentobarbitone, is a short-acting barbiturate. In high doses, pentobarbital causes death by respiratory arrest . Pentobarbital is a barbiturate (bar-BIT-chur-ate). Pentobarbital slows the activity of your brain and nervous system. Pentobarbital is used short-term as a sedative to treat insomnia, or to cause you to fall asleep for surgery. Pentobarbital is also used as an emergency treatment for seizures. When sodium pentobarbital, a barbiturate used often in single drug animal euthanasia, is administered in an overdose, it causes rapid unconsciousness followed by paralysis of the diaphragm. This drug may also kill via cardiac arrhythmia.